NMR evidence of the kinetic and thermodynamic products in the NIS promoted cyclization of 1-phenyl-4-pentenylamines. Synthesis and reactivity of trans-2-phenyl-5-iodopiperidines.

نویسندگان

  • Faïza Diaba
  • Josep Bonjoch
چکیده

The intramolecular reaction of secondary amines with tethered alkenes using NIS was studied, which gave insight into the kinetic vs. thermodynamic control of the iodoaminocyclization and the regioselectivity of the aziridinium ring-opening reactions, and led to functionalized piperidines.

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عنوان ژورنال:
  • Chemical communications

دوره 47 11  شماره 

صفحات  -

تاریخ انتشار 2011